Swiss-Prot entry
ID PXR_RAT STANDARD; PRT; 431 AA.
AC Q9R1A7;
DT 16-OCT-2001 (Rel. 40, Created)
DT 16-OCT-2001 (Rel. 40, Last sequence update)
DT 01-MAY-2005 (Rel. 47, Last annotation update)
DE Orphan nuclear receptor PXR (Pregnane X receptor).
GN Name=Nr1i2; Synonyms=Pxr;
OS Rattus norvegicus (Rat).
OC Eukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;
OC Mammalia; Eutheria; Euarchontoglires; Glires; Rodentia; Sciurognathi;
OC Muridae; Murinae; Rattus.
OX NCBI_TaxID=10116;
RN [1]
RP NUCLEOTIDE SEQUENCE.
RC STRAIN=Sprague-Dawley;
RX MEDLINE=99345883; PubMed=10415106 [NCBI, ExPASy, EBI, Israel, Japan]; DOI=10.1006/abbi.1999.1307;
RA Zhang H., LeCulyse E., Liu L., Hu M., Matoney L., Zhu W., Yan B.;
RT "Rat pregnane X receptor: molecular cloning, tissue distribution, and
RT xenobiotic regulation.";
RL Arch. Biochem. Biophys. 368:14-22(1999).
CC -!- FUNCTION: Orphan receptor; its natural ligand is probably
CC pregnane. Binds to a response element in CYP3A genes promoter (By
CC similarity).
CC -!- SUBUNIT: Forms a heterodimer with RXR (By similarity).
CC -!- SUBCELLULAR LOCATION: Nuclear (By similarity).
CC -!- SIMILARITY: Belongs to the nuclear hormone receptor family. NR1
CC subfamily.
CC -!- SIMILARITY: Contains 1 nuclear receptor DNA-binding domain.
CC --------------------------------------------------------------------------
CC This Swiss-Prot entry is copyright. It is produced through a collaboration
CC between the Swiss Institute of Bioinformatics and the EMBL outstation -
CC the European Bioinformatics Institute. There are no restrictions on its
CC use as long as its content is in no way modified and this statement is not
CC removed.
CC --------------------------------------------------------------------------
DR EMBL; AF151377; AAD47214.1; -. [EMBL / GenBank / DDBJ] [CoDingSequence]
DR HSSP; O75469; 1M13. [HSSP ENTRY / SWISS-3DIMAGE / PDB]
DR SMR; Q9R1A7; 139-429.
DR TRANSFAC; T04629; -.
DR Ensembl; ENSRNOG00000002906; Rattus_norvegicus
DR GO; GO:0004879; F:ligand-dependent nuclear receptor activity; IDA.
DR InterPro; IPR000536; Hrmon_recept_lig.
DR InterPro; IPR001723; Stdhrmn_receptor.
DR InterPro; IPR008946; Str_ncl_receptor.
DR InterPro; IPR000324; VitD_receptor.
DR InterPro; IPR001628; Znf_C4steroid.
DR InterPro; Graphical view of domain structure.
DR Pfam; PF00104; Hormone_recep; 1.
DR Pfam; PF00105; zf-C4; 1.
DR Pfam; Graphical view of domain structure.
DR PRINTS; PR00398; STRDHORMONER.
DR PRINTS; PR00047; STROIDFINGER.
DR PRINTS; PR00350; VITAMINDR.
DR ProDom; PD000035; Znf_C4steroid; 1.
DR ProDom [Domain structure / List of seq. sharing at least 1 domain ]
DR SMART; SM00430; HOLI; 1.
DR SMART; SM00399; ZnF_C4; 1.
DR PROSITE; PS00031; NUCLEAR_REC_DBD_1; 1.
DR PROSITE; PS51030; NUCLEAR_REC_DBD_2; 1.
DR CMR; Q9R1A7.
DR HOVERGEN [Family / Alignment / Tree]
DR BLOCKS; Q9R1A7.
DR ProtoNet; Q9R1A7.
DR ProtoMap; Q9R1A7.
DR PRESAGE; Q9R1A7.
DR DIP; Q9R1A7.
DR ModBase; Q9R1A7.
DR SWISS-2DPAGE; GET REGION ON 2D PAGE.
KW DNA-binding; Nuclear protein; Receptor; Transcription;
KW Transcription regulation; Zinc-finger.
FT DNA_BIND 38 104 Nuclear receptor-type.
FT ZN_FING 38 58 C4-type.
FT DOMAIN 63 89 Bipartite nuclear localization signal (By
FT similarity).
FT ZN_FING 74 99 C4-type.
FT DOMAIN 105 201 Hinge.
FT DOMAIN 202 431 Ligand-binding.
SQ SEQUENCE 431 AA; 49660 MW; 4B545F21F9439697 CRC64;
MRPEERWNHV GLVQREEADS VLEEPINVDE EDGGLQICRV CGDKANGYHF NVMTCEGCKG
FFRRAMKRNV RLRCPFRKGT CEITRKTRRQ CQACRLRKCL ESGMKKEMIM SDAAVEQRRA
LIKRKKREKI EAPPPGGQGL TEEQQALIQE LMDAQMQTFD TTFSHFKDFR LPAVFHSDCE
LPEVLQASLL EDPATWSQIM KDSVPMKISV QLRGEDGSIW NYQPPSKSDG KEIIPLLPHL
ADVSTYMFKG VINFAKVISH FRELPIEDQI SLLKGATFEM CILRFNTMFD TETGTWECGR
LAYCFEDPNG GFQKLLLDPL MKFHCMLKKL QLREEEYVLM QAISLFSPDR PGVVQRSVVD
QLQERFALTL KAYIECSRPY PAHRFLFLKI MAVLTELRSI NAQQTQQLLR IQDTHPFATP
LMQELFSSTD G
//