2005, NucleaRDB.
Each point mutation is linked to the entry specific to the residue position, Swiss-Prot ID to the list of mutations available for the corresponding protein, and Swiss-Prot AC to the table of cross-references. Citations are linked to the list of point mutations found in the corresponding articles. The putative locations of the point mutations are indicated in the second column and the corresponding general numbering in the third column, when appropriate.
Mutation Location Gl numbering Swiss-Prot ID (AC) Gene name Reference S16A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gioeli D et al.,2002 G21E N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Callewaert L et al.,2003 L26A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 He B et al.,2002 F27A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 He B et al.,2002 Q58L N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Lund A et al.,2003 S81A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gioeli D et al.,2002 S81A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Fu M et al.,2004 S81D N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gioeli D et al.,2002 S94A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gioeli D et al.,2002 S94A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Fu M et al.,2004 S119X N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 L121A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Liu Y et al.,2004 P151S N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Nesslinger NJ et al.,2003 D154N N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 LaFevre-Bernt MA et al.,2003 G166S N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Haapala K et al.,2001 L172X N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 S176S N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hyytinen ER et al.,2002 I182A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Alen P et al.,1999 I182A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Callewaert L et al.,2003 L183A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Alen P et al.,1999 L183A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Callewaert L et al.,2003 R210R N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Yan J et al.,2004 E211E N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Yan J et al.,2004 G214R N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Betney R et al.,2003 N222K N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Betney R et al.,2003 N233K N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Giwercman YL et al.,2001 N233K N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Lundin KB et al.,2003 N233K N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Holdcraft RW et al.,2004 S256A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gioeli D et al.,2002 S256A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Fu M et al.,2004 S308A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gioeli D et al.,2002 S308A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Fu M et al.,2004 S308D N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gioeli D et al.,2002 A355P N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Reid J et al.,2002 P390D N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hiort O et al.,2000 P390S N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hiort O et al.,2000 S424A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gioeli D et al.,2002 S424A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Fu M et al.,2004 S426A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Fu M et al.,2004 W433A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 He B et al.,2002 L436A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 He B et al.,2002 F437A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 He B et al.,2002 P514S N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hyytinen ER et al.,2002 P516S N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Yan J et al.,2004 K520E N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Liu GZ et al.,2003 G524A N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hyytinen ER et al.,2002 G524S N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hyytinen ER et al.,2002 D528G N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Liu GZ et al.,2003 P533S N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hyytinen ER et al.,2002 R538E N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Liu GZ et al.,2003 L547F N-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 C562G DNA_BIND D004 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Yen PM et al.,1997 G568V DNA_BIND D010 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Poukka H et al.,2000 L574P DNA_BIND D016 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 T575A DNA_BIND D017 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marcelli M et al.,2000 T575A DNA_BIND D017 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 S578T DNA_BIND D020 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Lundberg Giwercman Y et al.,2002 K580E DNA_BIND D022 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Liu GZ et al.,2003 K580R DNA_BIND D022 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marcelli M et al.,2000 K580R DNA_BIND D022 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 F582Y DNA_BIND D024 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Black BE et al.,2004 A586V DNA_BIND D028 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marcelli M et al.,2000 A586V DNA_BIND D028 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 A587S DNA_BIND D029 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marcelli M et al.,2000 A587S DNA_BIND D029 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 A596T DNA_BIND D038 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Lundberg Giwercman Y et al.,2002 A596T DNA_BIND D038 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Geserick C et al.,2003 S597R DNA_BIND D039 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Giwercman YL et al.,2003 R598D DNA_BIND D040 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Geserick C et al.,2003 T602P DNA_BIND D044 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 R607Q DNA_BIND D049 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Aarnisalo P et al.,1999 R607Q DNA_BIND D049 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Poukka H et al.,2000 R607X DNA_BIND D049 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Lundberg Giwercman Y et al.,2000 R608K DNA_BIND D050 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Aarnisalo P et al.,1999 R608K DNA_BIND D050 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Yeh S et al.,2003 R615G DNA_BIND D057 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Lundberg Giwercman Y et al.,2003 R617P DNA_BIND D059 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Heinlein CA et al.,2002 C619Y DNA_BIND D061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Nazareth LV et al.,1999 C619Y DNA_BIND D061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marcelli M et al.,2000 C619Y DNA_BIND D061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 C619Y DNA_BIND D061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Carsol JL et al.,2002 C619Y DNA_BIND D061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tan J et al.,1997 R629Q HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 K630A HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Fu M et al.,2000 K630A HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thomas M et al.,2004 K630A HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Fu M et al.,2004 K630Q HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Fu M et al.,2004 K630T HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 K632A HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Fu M et al.,2000 K632A HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thomas M et al.,2004 K633A HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Fu M et al.,2000 K633A HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thomas M et al.,2004 A645D HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Giwercman YL et al.,2002 A645D HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gottlieb B et al.,1997 S646F HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2003 S647N HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 T649T HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Segawa N et al.,2002 S650A HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gioeli D et al.,2002 S650A HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Fu M et al.,2004 S650D HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gioeli D et al.,2002 E653K HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Giwercman YL et al.,2002 I664N HINGE ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Giwercman YL et al.,2002 Q670R LBD HELIX 1 139 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 I672T LBD HELIX 1 141 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 P682T LBD HELIX 1 151 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Chavez B et al.,2002 G683A LBD HELIX 1 152 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 H689P Loop 1-3 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Rosa S et al.,2002 L701H LBD HELIX 3 332 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Zhao XY et al.,1999 L701H LBD HELIX 3 332 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Han G et al.,2001 L701H LBD HELIX 3 332 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 L701H LBD HELIX 3 332 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Chang CY et al.,2001 L701H LBD HELIX 3 332 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 L701H LBD HELIX 3 332 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Matias PM et al.,2002 L701H LBD HELIX 3 332 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Krishnan AV et al.,2002 L701H LBD HELIX 3 332 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hara T et al.,2003 L701H LBD HELIX 3 332 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ceraline J et al.,2003 L701H LBD HELIX 3 332 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Mooney SD et al.,2003 L701I LBD HELIX 3 332 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Chavez B et al.,2001 S703G LBD HELIX 3 334 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thin TH et al.,2002 N705A LBD HELIX 3 336 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marhefka CA et al.,2001 N705S LBD HELIX 3 336 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marhefka CA et al.,2001 N705S LBD HELIX 3 336 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thin TH et al.,2002 N705S LBD HELIX 3 336 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 L707R LBD HELIX 3 338 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marhefka CA et al.,2001 L707R LBD HELIX 3 338 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thin TH et al.,2002 G708A LBD HELIX 3 339 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Terouanne B et al.,2003 G708F LBD HELIX 3 339 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Terouanne B et al.,2003 G708V LBD HELIX 3 339 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Terouanne B et al.,2003 E709E LBD HELIX 3 340 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Segawa N et al.,2002 E709K LBD HELIX 3 340 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thin TH et al.,2002 Q711E LBD HELIX 3 342 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Chavez B et al.,2002 Q711E LBD HELIX 3 342 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thin TH et al.,2003 L712F LBD HELIX 3 343 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Holterhus PM et al.,2000 L712R LBD HELIX 3 343 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Alen P et al.,1999 V715A LBD HELIX 3 346 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Alen P et al.,1999 V715M LBD HELIX 3 346 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Taplin ME et al.,1999 V715M LBD HELIX 3 346 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 V715M LBD HELIX 3 346 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Grossmann ME et al.,2001 V715M LBD HELIX 3 346 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 V715M LBD HELIX 3 346 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hara T et al.,2003 V715M LBD HELIX 3 346 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tan J et al.,1997 V716A LBD HELIX 3 347 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Alen P et al.,1999 V716R LBD HELIX 3 347 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 He B et al.,2002 V716R LBD HELIX 3 347 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 K717E LBD HELIX 3 348 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 W718A LBD HELIX 3 349 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Alen P et al.,1999 A719K LBD HELIX 3 350 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Alen P et al.,1999 K720A LBD HELIX 3 351 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Alen P et al.,1999 K720A LBD HELIX 3 351 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 K720A LBD HELIX 3 351 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 He B et al.,2002 K720A LBD HELIX 3 351 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 K720A LBD HELIX 3 351 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Black BE et al.,2004 K720A LBD HELIX 3 351 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Alen P et al.,1999 K720E LBD HELIX 3 351 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 A721T LBD HELIX 3 352 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 G724D Loop 3-4 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 F725L Loop 3-4 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 F725L Loop 3-4 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ghali SA et al.,2003 R726L Loop 3-4 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Lim J et al.,2000 R726L Loop 3-4 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Mononen N et al.,2000 R726L Loop 3-4 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 R726L Loop 3-4 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 R726L Loop 3-4 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hyytinen ER et al.,2002 R726L Loop 3-4 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thin TH et al.,2003 R726L Loop 3-4 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gruber SB et al.,2003 R726L Loop 3-4 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Syrjakoski K et al.,2003 R726L Loop 3-4 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Koivisto PA et al.,2004 R726L Loop 3-4 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Yan J et al.,2004 N727K Loop 3-4 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Lim J et al.,2000 N727K Loop 3-4 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Wang Q et al.,2001 N727K Loop 3-4 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 N727K Loop 3-4 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ghali SA et al.,2003 V730M LBD HELIX 4 448 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 V730M LBD HELIX 4 448 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tan J et al.,1997 S740C LBD HELIX 4 458 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Pitteloud N et al.,2004 W741C LBD HELIX 5 548 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Haapala K et al.,2001 W741C LBD HELIX 5 548 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hara T et al.,2003 W741C LBD HELIX 5 548 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 W741L LBD HELIX 5 548 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hara T et al.,2003 W741R LBD HELIX 5 548 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 McPhaul MJ et al.,1999 W741R LBD HELIX 5 548 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marhefka CA et al.,2001 W741R LBD HELIX 5 548 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 McPhaul M et al.,2001 M742I LBD HELIX 5 549 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marhefka CA et al.,2001 M742V LBD HELIX 5 549 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marhefka CA et al.,2001 M742V LBD HELIX 5 549 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 M742V LBD HELIX 5 549 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ghali SA et al.,2003 M742V LBD HELIX 5 549 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 G743E LBD HELIX 5 550 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Chavez B et al.,2003 G743G LBD HELIX 5 550 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hyytinen ER et al.,2002 G743R LBD HELIX 5 550 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Chavez B et al.,2001 G743V LBD HELIX 5 550 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 G743V LBD HELIX 5 550 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gaughan L et al.,2001 L744L LBD HELIX 5 551 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hyytinen ER et al.,2002 M745T LBD HELIX 5 552 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marhefka CA et al.,2001 A748D LBD HELIX 5 555 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marcelli M et al.,2000 A748D LBD HELIX 5 555 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marhefka CA et al.,2001 A748T LBD HELIX 5 555 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 A748T LBD HELIX 5 555 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 James AJ et al.,2002 A748V LBD HELIX 5 555 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marcelli M et al.,2000 A748V LBD HELIX 5 555 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 M749I LBD HELIX 5 556 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Haapala K et al.,2001 M749I LBD HELIX 5 556 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 M749I LBD HELIX 5 556 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thin TH et al.,2003 M749L LBD HELIX 5 556 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thin TH et al.,2003 G750D LBD HELIX 5 557 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Bevan CL et al.,1997 G750S LBD HELIX 5 557 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 R752Q LBD HELIX 5 559 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Alen P et al.,1999 R752Q LBD HELIX 5 559 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marhefka CA et al.,2001 R752Q LBD HELIX 5 559 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Bubulya A et al.,2001 R752Q LBD HELIX 5 559 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Langley E et al.,1998 R752X LBD HELIX 5 559 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 F754L Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 F754L Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 T755A Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 N756S Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Giwercman YL et al.,2001 N756S Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Lundin KB et al.,2003 N756S Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Holdcraft RW et al.,2004 V757A Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marcelli M et al.,2000 V757A Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 V757I Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hyytinen ER et al.,2002 S759P Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 L762F Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Bevan CL et al.,1997 Y763C Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 Y763C Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 Y763C Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Murono K et al.,2003 Y763C Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Langley E et al.,1998 Y763H Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Langley E et al.,1998 F764L Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marhefka CA et al.,2001 A765S Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Chavez B et al.,2001 A765T Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Bevan CL et al.,1997 L768P Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 L768V Loop 5-6 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 E772A LBD HELIX 6 647 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ghali SA et al.,2003 E772A LBD HELIX 6 647 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gottlieb B et al.,1998 R774C LBD HELIX 6 649 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gottlieb B et al.,1998 R774C LBD HELIX 6 649 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 McPhaul MJ et al.,1999 R774C LBD HELIX 6 649 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 McPhaul M et al.,1999 R774C LBD HELIX 6 649 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ghali SA et al.,2003 R774C LBD HELIX 6 649 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Wu JH et al.,2003 R774C LBD HELIX 6 649 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Brown TR et al.,1990 R774H LBD HELIX 6 649 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gottlieb B et al.,1990 R779W Loop 6-7 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 R779W Loop 6-7 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Murono K et al.,2003 M780I Loop 6-7 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gottlieb B et al.,2003 M780I Loop 6-7 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Holterhus PM et al.,2000 S782N LBD HELIX 7 737 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 C784Y LBD HELIX 7 739 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 C784Y LBD HELIX 7 739 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Carsol JL et al.,2002 R786X LBD HELIX 7 741 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ignacak M et al.,2002 M787V LBD HELIX 7 742 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marhefka CA et al.,2001 S791P LBD HELIX 7 746 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 Q798E Loop 7-8 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hiort O et al.,2000 Q798E Loop 7-8 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 Q798E Loop 7-8 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Carsol JL et al.,2002 Q798E Loop 7-8 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Koivisto PA et al.,2004 P801T LBD HELIX 8 848 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 Q802R LBD HELIX 8 849 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Chavez B et al.,2001 F804L LBD HELIX 8 851 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gad YZ et al.,2003 M807R LBD HELIX 8 854 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ong YC et al.,2002 M807T LBD HELIX 8 854 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Loy CJ et al.,2001 M807T LBD HELIX 8 854 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ong YC et al.,2002 M807V LBD HELIX 8 854 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ong YC et al.,2002 M807V LBD HELIX 8 854 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 M807V LBD HELIX 8 854 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Murono K et al.,2003 L812F LBD HELIX 8 859 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Yaegashi N et al.,1999 L812F LBD HELIX 8 859 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Muroya K et al.,2001 S814N Loop 8-9 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ghali SA et al.,2003 P817A Loop 8-9 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Lumbroso S et al.,2004 Q824K LBD HELIX 9 936 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Giwercman A et al.,2000 F827V LBD HELIX 9 939 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Chavez B et al.,2000 L830P LBD HELIX 9 942 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 L830V LBD HELIX 9 942 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Chavez B et al.,2001 R831L LBD HELIX 9 943 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Chen CP et al.,2000 R831Q LBD HELIX 9 943 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gottlieb B et al.,2000 R831Q LBD HELIX 9 943 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Yaegashi N et al.,1999 R831Q LBD HELIX 9 943 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Chen CP et al.,2000 R831Q LBD HELIX 9 943 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Brown TR et al.,1990 R831X LBD HELIX 9 943 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Chen CP et al.,2000 R840C LBD HELIX 9 952 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,1999 R840C LBD HELIX 9 952 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Mazen I et al.,2004 R840G LBD HELIX 9 952 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,1999 R840G LBD HELIX 9 952 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Mazen I et al.,2004 R840H LBD HELIX 9 952 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,1999 R840H LBD HELIX 9 952 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Mazen I et al.,2004 R840S LBD HELIX 9 952 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 R840S LBD HELIX 9 952 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Mazen I et al.,2004 R846G LBD HELIX 9 958 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marcelli M et al.,2000 R846G LBD HELIX 9 958 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 R846H LBD HELIX 9 958 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Boehmer AL et al.,2001 R855C LBD HELIX 10-11 1039 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 R855C LBD HELIX 10-11 1039 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Elhaji YA et al.,2004 R855C LBD HELIX 10-11 1039 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Murono K et al.,2004 R855H LBD HELIX 10-11 1039 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 R855H LBD HELIX 10-11 1039 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Elhaji YA et al.,2004 D864N LBD HELIX 10-11 1048 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Bevan CL et al.,1997 S865P LBD HELIX 10-11 1049 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marcelli M et al.,2000 S865P LBD HELIX 10-11 1049 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 V866M LBD HELIX 10-11 1050 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 V866M LBD HELIX 10-11 1050 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hyytinen ER et al.,2002 V866M LBD HELIX 10-11 1050 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ghali SA et al.,2003 V866M LBD HELIX 10-11 1050 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Brown TR et al.,1990 V866M LBD HELIX 10-11 1050 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Langley E et al.,1998 A870E LBD HELIX 10-11 1054 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Chen CP et al.,2000 R871G LBD HELIX 10-11 1055 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ghali SA et al.,2003 R871G LBD HELIX 10-11 1055 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gottlieb B et al.,1998 H874R LBD HELIX 10-11 1058 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Chavez B et al.,1998 H874Y LBD HELIX 10-11 1058 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Taplin ME et al.,1999 H874Y LBD HELIX 10-11 1058 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 McDonald S et al.,2000 H874Y LBD HELIX 10-11 1058 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Grossmann ME et al.,2001 H874Y LBD HELIX 10-11 1058 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 H874Y LBD HELIX 10-11 1058 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Solit DB et al.,2002 H874Y LBD HELIX 10-11 1058 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Steketee K et al.,2002 H874Y LBD HELIX 10-11 1058 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thin TH et al.,2003 H874Y LBD HELIX 10-11 1058 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hara T et al.,2003 H874Y LBD HELIX 10-11 1058 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shao TC et al.,2003 H874Y LBD HELIX 10-11 1058 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tan J et al.,1997 T877 LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Buchanan G et al.,2001 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Taplin ME et al.,1999 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Zhao XY et al.,1999 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 McDonald S et al.,2000 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Truica CI et al.,2000 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Han G et al.,2001 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Kang HY et al.,2001 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Sack JS et al.,2001 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marhefka CA et al.,2001 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tomura A et al.,2001 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Grossmann ME et al.,2001 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Haapala K et al.,2001 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Chang CY et al.,2001 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Matias PM et al.,2002 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Krishnan AV et al.,2002 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Solit DB et al.,2002 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Cheng S et al.,2002 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Steketee K et al.,2002 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Maggiolini M et al.,2002 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hyytinen ER et al.,2002 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thin TH et al.,2003 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hara T et al.,2003 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ceraline J et al.,2003 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Berrevoets CA et al.,2002 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Rahman MM et al.,2003 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Mooney SD et al.,2003 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Rahman MM et al.,2003 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ghali SA et al.,2003 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ishioka T et al.,2003 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2003 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ceraline J et al.,2004 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gregory CW et al.,2004 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ai N et al.,2003 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Berrevoets CA et al.,2004 T877A LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gottlieb B et al.,1997 T877C LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Steketee K et al.,2002 T877G LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Steketee K et al.,2002 T877S LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Taplin ME et al.,1999 T877S LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Steketee K et al.,2002 T877S LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thin TH et al.,2003 T877S LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Hara T et al.,2003 T877S LBD HELIX 10-11 1061 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tan J et al.,1997 D879Y Loop 11-12 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Chavez B et al.,1997 L880Q Loop 11-12 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 M886V Loop 11-12 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ghadessy FJ et al.,1999 M886V Loop 11-12 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Lim J et al.,2000 M886V Loop 11-12 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Wang Q et al.,2001 M886V Loop 11-12 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 M886V Loop 11-12 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ghali SA et al.,2003 S888S Loop 11-12 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Chavez B et al.,2003 V889M Loop 11-12 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ghadessy FJ et al.,1999 V889M Loop 11-12 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Alen P et al.,1999 V889M Loop 11-12 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marhefka CA et al.,2001 V889M Loop 11-12 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Bubulya A et al.,2001 V889M Loop 11-12 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 V889M Loop 11-12 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Langley E et al.,1998 D890N Loop 11-12 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Taplin ME et al.,1999 D890N Loop 11-12 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 F891A Loop 11-12 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 F891L Loop 11-12 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Gottlieb B et al.,2003 F891L Loop 11-12 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 P892L LBD HELIX 12 1245 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 E893A LBD HELIX 12 1246 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 M894A LBD HELIX 12 1247 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Slagsvold T et al.,2000 M894A LBD HELIX 12 1247 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 M894A LBD HELIX 12 1247 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 M894D LBD HELIX 12 1247 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Slagsvold T et al.,2000 M894D LBD HELIX 12 1247 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 M894D LBD HELIX 12 1247 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 M895A LBD HELIX 12 1248 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Slagsvold T et al.,2000 M895A LBD HELIX 12 1248 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 M895T LBD HELIX 12 1248 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marhefka CA et al.,2001 M895T LBD HELIX 12 1248 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 M895T LBD HELIX 12 1248 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 A896L LBD HELIX 12 1249 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 A896T LBD HELIX 12 1249 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 A896V LBD HELIX 12 1249 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Slagsvold T et al.,2000 A896V LBD HELIX 12 1249 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 A896V LBD HELIX 12 1249 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 E897K LBD HELIX 12 1250 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 He B et al.,2002 E897Q LBD HELIX 12 1250 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Ghadessy FJ et al.,1999 E897V LBD HELIX 12 1250 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Slagsvold T et al.,2000 E897V LBD HELIX 12 1250 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 I898A LBD HELIX 12 1251 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Alen P et al.,1999 I898A LBD HELIX 12 1251 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 I898F LBD HELIX 12 1251 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 I898T LBD HELIX 12 1251 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 I898T LBD HELIX 12 1251 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 I899A LBD HELIX 12 1252 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Alen P et al.,1999 I899A LBD HELIX 12 1252 ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 Q902R C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 Q902R C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 V903M C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 V903M C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 P904H C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 P904H C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 P904R C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 P904S C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 P904S C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 P904S C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 P904V C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Melo KF et al.,2003 K905A C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 L907A C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tahiri B et al.,2001 L907F C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Thompson J et al.,2001 L907F C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 L907F C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Bevan CL et al.,1997 G909A C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tahiri B et al.,2001 G909E C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tahiri B et al.,2001 G909E C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 G909R C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Song LN et al.,2003 K910A C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tahiri B et al.,2001 K910R C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 V911G C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tahiri B et al.,2001 K912A C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tahiri B et al.,2001 I914A C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tahiri B et al.,2001 Y915A C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tahiri B et al.,2001 F916A C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tahiri B et al.,2001 F916P C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tahiri B et al.,2001 F916Y C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tahiri B et al.,2001 H917A C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tahiri B et al.,2001 H917R C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Sack JS et al.,2001 Q919C C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tahiri B et al.,2001 Q919R C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Marcelli M et al.,2000 Q919R C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tahiri B et al.,2001 Q919R C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Shi XB et al.,2002 Q919R C-term ANDR_HUMAN (P10275) AR,DHTR, NR3C4 Tan J et al.,1997 P140P N-term ANDR_MOUSE (P19091) Ar,Nr3c4 Han G et al.,2001 E206K N-term ANDR_MOUSE (P19091) Ar,Nr3c4 Han G et al.,2001 A229T N-term ANDR_MOUSE (P19091) Ar,Nr3c4 Han G et al.,2001 E231G N-term ANDR_MOUSE (P19091) Ar,Nr3c4 Han G et al.,2001 E231G N-term ANDR_MOUSE (P19091) Ar,Nr3c4 Culig Z et al.,2001 R273C N-term ANDR_MOUSE (P19091) Ar,Nr3c4 Nesslinger NJ et al.,2003 R273H N-term ANDR_MOUSE (P19091) Ar,Nr3c4 Nesslinger NJ et al.,2003 N384S N-term ANDR_MOUSE (P19091) Ar,Nr3c4 Han G et al.,2001 A394A N-term ANDR_MOUSE (P19091) Ar,Nr3c4 Han G et al.,2001 V487A N-term ANDR_MOUSE (P19091) Ar,Nr3c4 Han G et al.,2001 K638M HINGE ANDR_MOUSE (P19091) Ar,Nr3c4 Han G et al.,2001 F653 LBD HELIX 1 142 ANDR_MOUSE (P19091) Ar,Nr3c4 Buchanan G et al.,2001 F653F LBD HELIX 1 142 ANDR_MOUSE (P19091) Ar,Nr3c4 Han G et al.,2001 F653I LBD HELIX 1 142 ANDR_MOUSE (P19091) Ar,Nr3c4 Han G et al.,2001 S676S Loop 1-3 ANDR_MOUSE (P19091) Ar,Nr3c4 Han G et al.,2001 F677S LBD HELIX 3 328 ANDR_MOUSE (P19091) Ar,Nr3c4 Han G et al.,2001 R754H LBD HELIX 6 649 ANDR_MOUSE (P19091) Ar,Nr3c4 Han G et al.,2001 D844D LBD HELIX 10-11 1048 ANDR_MOUSE (P19091) Ar,Nr3c4 Han G et al.,2001 T857A LBD HELIX 10-11 1061 ANDR_MOUSE (P19091) Ar,Nr3c4 Han G et al.,2001 E877G LBD HELIX 12 1250 ANDR_MOUSE (P19091) Ar,Nr3c4 Han G et al.,2001 I163N N-term ANDR_RAT (P15207) Ar,Nr3c4 Chamberlain NL et al.,1996 L164N N-term ANDR_RAT (P15207) Ar,Nr3c4 Chamberlain NL et al.,1996 S165A N-term ANDR_RAT (P15207) Ar,Nr3c4 Chamberlain NL et al.,1996 S340A N-term ANDR_RAT (P15207) Ar,Nr3c4 Reid J et al.,2002 A353P N-term ANDR_RAT (P15207) Ar,Nr3c4 Reid J et al.,2002 S514A N-term ANDR_RAT (P15207) Ar,Nr3c4 LaFevre-Bernt MA et al.,2003 G551V DNA_BIND D010 ANDR_RAT (P15207) Ar,Nr3c4 Aarnisalo P et al.,1999 G551V DNA_BIND D010 ANDR_RAT (P15207) Ar,Nr3c4 Poukka H et al.,2000 C552A DNA_BIND D011 ANDR_RAT (P15207) Ar,Nr3c4 Shaffer PL et al.,2004 C562G DNA_BIND D021 ANDR_RAT (P15207) Ar,Nr3c4 Aarnisalo P et al.,1999 C562G DNA_BIND D021 ANDR_RAT (P15207) Ar,Nr3c4 Poukka H et al.,2000 K563A DNA_BIND D022 ANDR_RAT (P15207) Ar,Nr3c4 Aarnisalo P et al.,1999 K563A DNA_BIND D022 ANDR_RAT (P15207) Ar,Nr3c4 Poukka H et al.,2000 A579T DNA_BIND D038 ANDR_RAT (P15207) Ar,Nr3c4 Aarnisalo P et al.,1999 A579T DNA_BIND D038 ANDR_RAT (P15207) Ar,Nr3c4 Poukka H et al.,2000 A579T DNA_BIND D038 ANDR_RAT (P15207) Ar,Nr3c4 Shaffer PL et al.,2004 S580T DNA_BIND D039 ANDR_RAT (P15207) Ar,Nr3c4 Shaffer PL et al.,2004 R581D DNA_BIND D040 ANDR_RAT (P15207) Ar,Nr3c4 Chen S et al.,1997 T585A DNA_BIND D044 ANDR_RAT (P15207) Ar,Nr3c4 Shaffer PL et al.,2004 R590Q DNA_BIND D049 ANDR_RAT (P15207) Ar,Nr3c4 Aarnisalo P et al.,1999 R590Q DNA_BIND D049 ANDR_RAT (P15207) Ar,Nr3c4 Poukka H et al.,2000 C597G DNA_BIND D056 ANDR_RAT (P15207) Ar,Nr3c4 Poukka H et al.,2000 R600G DNA_BIND D059 ANDR_RAT (P15207) Ar,Nr3c4 Poukka H et al.,2000 K601A DNA_BIND D060 ANDR_RAT (P15207) Ar,Nr3c4 Poukka H et al.,2000 Y603C DNA_BIND D062 ANDR_RAT (P15207) Ar,Nr3c4 Poukka H et al.,2000 Y81X N-term DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Zhang YH et al.,2001 Q224A N-term DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Lehmann SG et al.,2002 R267A LBD HELIX 3 348 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Lalli E et al.,2000 R267A LBD HELIX 3 348 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Lehmann SG et al.,2002 R267A LBD HELIX 3 348 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Lalli E et al.,1997 R267P LBD HELIX 3 348 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Altincicek B et al.,2000 R267P LBD HELIX 3 348 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Lalli E et al.,2000 R267P LBD HELIX 3 348 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Achermann JC et al.,2001 R267P LBD HELIX 3 348 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Holter E et al.,2002 R267P LBD HELIX 3 348 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Lehmann SG et al.,2002 R267P LBD HELIX 3 348 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Ito M et al.,1997 R267P LBD HELIX 3 348 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Lalli E et al.,1997 V269A LBD HELIX 3 350 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Lalli E et al.,1997 R288A LBD HELIX 4 456 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Lehmann SG et al.,2002 L295P LBD HELIX 5 552 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Zhang YH et al.,2001 A300P LBD HELIX 5 557 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Achermann JC et al.,2001 A300V LBD HELIX 5 557 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Achermann JC et al.,2001 E377K LBD HELIX 8 850 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Achermann JC et al.,2001 Y380D LBD HELIX 8 853 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Mantovani G et al.,2002 L381H LBD HELIX 8 854 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Mantovani G et al.,2002 R425G LBD HELIX 10-11 1039 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Achermann JC et al.,2001 R425T LBD HELIX 10-11 1039 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Achermann JC et al.,2001 R425T LBD HELIX 10-11 1039 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Zhang YH et al.,2001 E428X LBD HELIX 10-11 1042 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Zhang YH et al.,2001 I439S LBD HELIX 10-11 1053 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Achermann JC et al.,2001 I439S LBD HELIX 10-11 1053 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Mantovani G et al.,2002 I439S LBD HELIX 10-11 1053 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Lehmann SG et al.,2002 N440A LBD HELIX 10-11 1054 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Lehmann SG et al.,2002 N440I LBD HELIX 10-11 1054 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Lalli E et al.,2000 N440I LBD HELIX 10-11 1054 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Lehmann SG et al.,2002 F449D Loop 11-12 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Achermann JC et al.,2001 M461A LBD HELIX 12 1247 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Lehmann SG et al.,2002 M462A LBD HELIX 12 1248 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Lehmann SG et al.,2002 E464R LBD HELIX 12 1250 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Lehmann SG et al.,2002 M465A LBD HELIX 12 1251 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Lehmann SG et al.,2002 L466A LBD HELIX 12 1252 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Lehmann SG et al.,2002 L466R LBD HELIX 12 1252 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Achermann JC et al.,2001 L466R LBD HELIX 12 1252 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Lehmann SG et al.,2002 L466R LBD HELIX 12 1252 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Mizusaki H et al.,2003 L466R LBD HELIX 12 1252 DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Kawajiri K et al.,2003 C467S C-term DAX1_HUMAN (P51843) NR0B1,AHC, DAX1 Achermann JC et al.,2001 M464A LBD HELIX 12 1248 DAX1_MOUSE (Q61066) Nr0b1,Ahch, Dax1 Kawajiri K et al.,2003 E466A LBD HELIX 12 1250 DAX1_MOUSE (Q61066) Nr0b1,Ahch, Dax1 Kawajiri K et al.,2003 L468A LBD HELIX 12 1252 DAX1_MOUSE (Q61066) Nr0b1,Ahch, Dax1 Kawajiri K et al.,2003 C469A C-term DAX1_MOUSE (Q61066) Nr0b1,Ahch, Dax1 Kawajiri K et al.,2003 L353R LBD HELIX 10-11 1043 EAR2_HUMAN (P10588) NR2F6,EAR2, ERBAL2 DeLong LJ et al.,2004 L360R LBD HELIX 10-11 1050 EAR2_HUMAN (P10588) NR2F6,EAR2, ERBAL2 DeLong LJ et al.,2004 C300Y DNA_BIND D037 ECR_DROME (P34021) EcR,NR1H1,CG1765 Gates J et al.,2004 R344Q HINGE ECR_DROME (P34021) EcR,NR1H1,CG1765 Carney GE et al.,2000 E476 LBD HELIX 3 348 ECR_DROME (P34021) EcR,NR1H1,CG1765 Grebe M et al.,2003 A483T Loop 3-4 ECR_DROME (P34021) EcR,NR1H1,CG1765 Carney GE et al.,2000 K497 LBD HELIX 4 456 ECR_DROME (P34021) EcR,NR1H1,CG1765 Grebe M et al.,2003 M504 LBD HELIX 5 552 ECR_DROME (P34021) EcR,NR1H1,CG1765 Grebe M et al.,2003 R511 LBD HELIX 5 559 ECR_DROME (P34021) EcR,NR1H1,CG1765 Grebe M et al.,2003 D572 Loop 8-9 ECR_DROME (P34021) EcR,NR1H1,CG1765 Grebe M et al.,2003 A612 LBD HELIX 10-11 1041 ECR_DROME (P34021) EcR,NR1H1,CG1765 Grebe M et al.,2003 L615 LBD HELIX 10-11 1044 ECR_DROME (P34021) EcR,NR1H1,CG1765 Grebe M et al.,2003 I617 LBD HELIX 10-11 1046 ECR_DROME (P34021) EcR,NR1H1,CG1765 Grebe M et al.,2003 T619 LBD HELIX 10-11 1048 ECR_DROME (P34021) EcR,NR1H1,CG1765 Grebe M et al.,2003 N626 LBD HELIX 10-11 1055 ECR_DROME (P34021) EcR,NR1H1,CG1765 Grebe M et al.,2003 F645A LBD HELIX 12 1247 ECR_DROME (P34021) EcR,NR1H1,CG1765 Cherbas L et al.,2003 F645A LBD HELIX 12 1247 ECR_DROME (P34021) EcR,NR1H1,CG1765 Hu X et al.,2003 E648 LBD HELIX 12 1250 ECR_DROME (P34021) EcR,NR1H1,CG1765 Grebe M et al.,2003 W650A LBD HELIX 12 1252 ECR_DROME (P34021) EcR,NR1H1,CG1765 Cherbas L et al.,2003 W650A LBD HELIX 12 1252 ECR_DROME (P34021) EcR,NR1H1,CG1765 Hu X et al.,2003 S73A N-term ERR1_HUMAN (P11474) ESRRA,ERR1, ESRL1, NR3B1 Qi X et al.,2004 S124A N-term ERR1_HUMAN (P11474) ESRRA,ERR1, ESRL1, NR3B1 Dutertre M et al.,2003 E129K N-term ERR1_HUMAN (P11474) ESRRA,ERR1, ESRL1, NR3B1 Oxelmark E et al.,2003 K201A DNA_BIND D026 ERR1_HUMAN (P11474) ESRRA,ERR1, ESRL1, NR3B1 Kim K et al.,2003 E390Q LBD HELIX 6 647 ERR1_HUMAN (P11474) ESRRA,ERR1, ESRL1, NR3B1 Stoica A et al.,2000 Y365M LBD HELIX 8 851 ERR1_MOUSE (O08580) Esrra,Err1, Estrra, Nr3b1 Ostberg T et al.,2003 L398A LBD HELIX 9 950 ERR1_MOUSE (O08580) Esrra,Err1, Estrra, Nr3b1 Huppunen J et al.,2004 E413A Loop 9-10 ERR1_MOUSE (O08580) Esrra,Err1, Estrra, Nr3b1 Huppunen J et al.,2004 S136A DNA_BIND D009 ERR3_HUMAN (P62508) ESRRG,ERR3, ERRG2, KIAA0832, NR3B3 Fernando RI et al.,2004 A272F LBD HELIX 3 339 ERR3_HUMAN (P62508) ESRRG,ERR3, ERRG2, KIAA0832, NR3B3 Greschik H et al.,2002 A272F LBD HELIX 3 339 ERR3_HUMAN (P62508) ESRRG,ERR3, ERRG2, KIAA0832, NR3B3 Huppunen J et al.,2004 A272L LBD HELIX 3 339 ERR3_HUMAN (P62508) ESRRG,ERR3, ERRG2, KIAA0832, NR3B3 Greschik H et al.,2002 L345I LBD HELIX 7 738 ERR3_HUMAN (P62508) ESRRG,ERR3, ERRG2, KIAA0832, NR3B3 Greschik H et al.,2002 F435L LBD HELIX 10-11 1061 ERR3_HUMAN (P62508) ESRRG,ERR3, ERRG2, KIAA0832, NR3B3 Greschik H et al.,2002 H6Y N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Feng J et al.,2001 A13V N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Oxelmark E et al.,2003 S104A N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Martin MB et al.,2000 S104A N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Coleman KM et al.,2003 S104A N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Dutertre M et al.,2003 S106A N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Martin MB et al.,2000 S106A N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Dutertre M et al.,2003 S118 N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen D et al.,2002 S118 N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Kato S et al.,1995 S118A N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Webb P et al.,1999 S118A N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Martin MB et al.,2000 S118A N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Lu D et al.,2001 S118A N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Singleton DW et al.,2003 S118A N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Dutertre M et al.,2003 S118A N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Deblois G et al.,2003 S118A N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 El-Tanani MK et al.,1997 S118E N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Webb P et al.,1999 S118E N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Dutertre M et al.,2003 S118R N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Webb P et al.,1999 P146Q N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Feng J et al.,2001 S167A N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Martin MB et al.,2000 S167A N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Clark DE et al.,2001 S167A N-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Sun M et al.,2001 C202H DNA_BIND D018 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Mize AL et al.,2003 C202R DNA_BIND D018 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 MacGregor Schafer J et al.,2001 E203G DNA_BIND D019 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Platet N et al.,2000 E203V DNA_BIND D019 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 MacGregor Schafer J et al.,2001 C205H DNA_BIND D021 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Mize AL et al.,2003 A207V DNA_BIND D023 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Platet N et al.,2000 S236A DNA_BIND D052 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Coleman KM et al.,2003 K299R HINGE ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Feng J et al.,2001 K299R HINGE ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Eng FC et al.,1997 K302A HINGE ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Garcia Pedrero JM et al.,2002 K302G HINGE ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Garcia Pedrero JM et al.,2002 K303A HINGE ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Garcia Pedrero JM et al.,2002 K303G HINGE ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Garcia Pedrero JM et al.,2002 K303R HINGE ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Fuqua SA et al.,2000 K303R HINGE ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Mishra SK et al.,2003 K303R HINGE ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Tokunaga E et al.,2004 S305A HINGE ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Wang RA et al.,2002 S305A HINGE ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Coleman KM et al.,2003 S305A HINGE ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Balasenthil S et al.,2004 S305E HINGE ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Wang RA et al.,2002 S305E HINGE ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Balasenthil S et al.,2004 T311A LBD HELIX 1 138 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Lee H et al.,2002 P325P LBD HELIX 1 152 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Bitenc D et al.,2001 P325P LBD HELIX 1 152 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Jurada S et al.,2001 S338A Loop 1-3 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Coleman KM et al.,2003 L349 LBD HELIX 3 338 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Matthews JB et al.,2001 D351A LBD HELIX 3 340 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Anghel SI et al.,2000 D351E LBD HELIX 3 340 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Anghel SI et al.,2000 D351G LBD HELIX 3 340 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Anghel SI et al.,2000 D351G LBD HELIX 3 340 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Bentrem D et al.,2001 D351G LBD HELIX 3 340 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Levenson AS et al.,2003 D351G LBD HELIX 3 340 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Mishra SK et al.,2003 D351G LBD HELIX 3 340 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Gehm BD et al.,2004 D351R LBD HELIX 3 340 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Mishra SK et al.,2003 D351V LBD HELIX 3 340 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Anghel SI et al.,2000 D351Y LBD HELIX 3 340 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Anghel SI et al.,2000 D351Y LBD HELIX 3 340 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Yao K et al.,2000 D351Y LBD HELIX 3 340 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Webb P et al.,2000 D351Y LBD HELIX 3 340 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Bentrem D et al.,2001 D351Y LBD HELIX 3 340 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Liu H et al.,2001 D351Y LBD HELIX 3 340 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Yamamoto Y et al.,2001 D351Y LBD HELIX 3 340 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Levenson AS et al.,2003 D351Y LBD HELIX 3 340 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Mishra SK et al.,2003 D351Y LBD HELIX 3 340 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Yamamoto Y et al.,2003 E353A LBD HELIX 3 342 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2003 E353Q LBD HELIX 3 342 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2004 I358F LBD HELIX 3 347 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2003 I358R LBD HELIX 3 347 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Yamamoto Y et al.,2001 K362A LBD HELIX 3 351 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Webb P et al.,1999 K362A LBD HELIX 3 351 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Webb P et al.,2000 K362A LBD HELIX 3 351 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Marimuthu A et al.,2002 K362A LBD HELIX 3 351 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Weatherman RV et al.,2002 K362A LBD HELIX 3 351 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Webb P et al.,2003 K362E LBD HELIX 3 351 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2003 G366T Loop 3-4 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Yamamoto Y et al.,2001 T371R LBD HELIX 4 447 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Webb P et al.,2003 D374N LBD HELIX 4 450 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Pakdel F et al.,1993 V376R LBD HELIX 4 452 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Webb P et al.,2000 V376R LBD HELIX 4 452 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Yamamoto Y et al.,2001 V376R LBD HELIX 4 452 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Webb P et al.,2003 L379R LBD HELIX 4 455 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Webb P et al.,2003 E380G LBD HELIX 4 456 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Ko L et al.,2002 E380Q LBD HELIX 4 456 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 E380Q LBD HELIX 4 456 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Pakdel F et al.,1993 E380Q LBD HELIX 4 456 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Lazennec G et al.,1997 C381 LBD HELIX 4 457 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Katzenellenbogen BS et al.,1993 C381A LBD HELIX 4 457 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 C381A LBD HELIX 4 457 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 C381S LBD HELIX 4 457 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Renaud J et al.,2003 C381S LBD HELIX 4 457 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Hurth KM et al.,2004 L384M LBD HELIX 5 549 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Sun J et al.,2003 E385Q LBD HELIX 5 550 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Pakdel F et al.,1993 I386P LBD HELIX 5 551 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2003 G390D LBD HELIX 5 555 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2004 G400V Loop 5-6 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Knoblauch R et al.,1999 G400V Loop 5-6 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Anghel SI et al.,2000 G400V Loop 5-6 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Webb P et al.,2000 G400V Loop 5-6 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Teyssier C et al.,2001 G400V Loop 5-6 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Webb P et al.,2003 G400V Loop 5-6 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Leone DP et al.,2003 G400V Loop 5-6 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Oxelmark E et al.,2003 G400V Loop 5-6 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Ramkumar T et al.,1995 G400V Loop 5-6 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Lee HS et al.,1996 G400V Loop 5-6 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Aumais JP et al.,1997 G400V Loop 5-6 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 El-Tanani MK et al.,1997 G400V Loop 5-6 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Eng FC et al.,1997 G400V Loop 5-6 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Logie C et al.,1998 K416Q LBD HELIX 6 651 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Pakdel F et al.,1993 C417A LBD HELIX 6 652 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 C417A LBD HELIX 6 652 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 C417S LBD HELIX 6 652 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Renaud J et al.,2003 C417S LBD HELIX 6 652 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Hurth KM et al.,2004 V422M LBD HELIX 7 736 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2003 G442E LBD HELIX 8 848 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2004 G442E LBD HELIX 8 848 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Eng FC et al.,1997 G442V LBD HELIX 8 848 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2004 C447A LBD HELIX 8 853 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 C447A LBD HELIX 8 853 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 C447A LBD HELIX 8 853 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Acconcia F et al.,2004 T460A Loop 8-9 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2003 F461I Loop 8-9 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2004 T465P Loop 8-9 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Eng FC et al.,1997 H501R Loop 9-10 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2003 R503A LBD HELIX 10-11 1039 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Logie C et al.,1998 L507R LBD HELIX 10-11 1043 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Logie C et al.,1998 L508R LBD HELIX 10-11 1044 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Nichols M et al.,1998 H516A LBD HELIX 10-11 1052 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Aliau S et al.,2002 S518A LBD HELIX 10-11 1054 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Wang RA et al.,2002 S518A LBD HELIX 10-11 1054 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Coleman KM et al.,2003 G521R LBD HELIX 10-11 1057 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Werdien D et al.,2001 G521R LBD HELIX 10-11 1057 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Preisler-Mashek MT et al.,2002 G521R LBD HELIX 10-11 1057 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Roscilli G et al.,2002 G521R LBD HELIX 10-11 1057 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Nichols M et al.,1998 G521R LBD HELIX 10-11 1057 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Schwenk F et al.,1998 G521R LBD HELIX 10-11 1057 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Logie C et al.,1998 G521V LBD HELIX 10-11 1057 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Logie C et al.,1998 E523A LBD HELIX 10-11 1059 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 E523A LBD HELIX 10-11 1059 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 E523Q LBD HELIX 10-11 1059 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 E523Q LBD HELIX 10-11 1059 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 H524A LBD HELIX 10-11 1060 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 H524A LBD HELIX 10-11 1060 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 H524A LBD HELIX 10-11 1060 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Aliau S et al.,2002 L525A LBD HELIX 10-11 1061 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Aliau S et al.,2002 M528 Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Matthews JB et al.,2001 K529Q Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 C530 Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Katzenellenbogen BS et al.,1993 C530A Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 C530A Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 C530S Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Renaud J et al.,2003 C530S Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Hurth KM et al.,2004 C530W Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Scarlata S et al.,1995 K531Q Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 N532D Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 L536A Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Zhao C et al.,2003 L536A Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2004 L536E Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Zhao C et al.,2003 L536E Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2004 L536G Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Zhao C et al.,2003 L536H Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2004 L536I Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Zhao C et al.,2003 L536K Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Zhao C et al.,2003 L536K Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2004 L536N Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Zhao C et al.,2003 L536N Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2004 L536P Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Anghel SI et al.,2000 L536P Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Zhao C et al.,2003 L536P Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2004 L536P Loop 11-12 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Eng FC et al.,1997 Y537A LBD HELIX 12 1245 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Anghel SI et al.,2000 Y537A LBD HELIX 12 1245 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Weis KE et al.,1996 Y537A LBD HELIX 12 1245 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Lazennec G et al.,1997 Y537E LBD HELIX 12 1245 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Zhong L et al.,2002 Y537E LBD HELIX 12 1245 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Weis KE et al.,1996 Y537F LBD HELIX 12 1245 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Zhong L et al.,2002 Y537F LBD HELIX 12 1245 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Arnold SF et al.,1995 Y537F LBD HELIX 12 1245 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Arnold SF et al.,1997 Y537K LBD HELIX 12 1245 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Weis KE et al.,1996 Y537N LBD HELIX 12 1245 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Fuqua SA et al.,2000 Y537N LBD HELIX 12 1245 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Zhong L et al.,2002 Y537N LBD HELIX 12 1245 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Eng FC et al.,1998 Y537S LBD HELIX 12 1245 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Zhong L et al.,2002 Y537S LBD HELIX 12 1245 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Weis KE et al.,1996 Y537S LBD HELIX 12 1245 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Eng FC et al.,1997 Y537S LBD HELIX 12 1245 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Lazennec G et al.,1997 D538A LBD HELIX 12 1246 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Liu H et al.,2001 D538A LBD HELIX 12 1246 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Sathya G et al.,2002 D538A LBD HELIX 12 1246 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Pearce ST et al.,2003 D538A LBD HELIX 12 1246 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Gehm BD et al.,2004 D538N LBD HELIX 12 1246 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Tcherepanova I et al.,2000 D538N LBD HELIX 12 1246 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 D538N LBD HELIX 12 1246 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Stoica A et al.,2000 D538N LBD HELIX 12 1246 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Saville B et al.,2002 D538N LBD HELIX 12 1246 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Kim K et al.,2003 D538N LBD HELIX 12 1246 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Norris JD et al.,1998 L539A LBD HELIX 12 1247 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Pearce ST et al.,2003 L539A LBD HELIX 12 1247 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Bai Y et al.,2003 L539A LBD HELIX 12 1247 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Deblois G et al.,2003 L540A LBD HELIX 12 1248 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Pearce ST et al.,2003 L540P LBD HELIX 12 1248 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Nichols M et al.,1998 L540Q LBD HELIX 12 1248 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Delage-Mourroux R et al.,2000 L540Q LBD HELIX 12 1248 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Pearce ST et al.,2003 L540Q LBD HELIX 12 1248 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Zhao C et al.,2003 L540Q LBD HELIX 12 1248 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Acevedo ML et al.,2004 L540Q LBD HELIX 12 1248 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Ince BA et al.,1995 L540Q LBD HELIX 12 1248 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Nichols M et al.,1998 E542A LBD HELIX 12 1250 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Liu H et al.,2001 E542A LBD HELIX 12 1250 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Sathya G et al.,2002 E542A LBD HELIX 12 1250 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Pearce ST et al.,2003 E542A LBD HELIX 12 1250 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Gehm BD et al.,2004 E542K LBD HELIX 12 1250 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Webb P et al.,2000 E542K LBD HELIX 12 1250 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Webb P et al.,2003 E542N LBD HELIX 12 1250 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Tcherepanova I et al.,2000 E542Q LBD HELIX 12 1250 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Saville B et al.,2002 E542Q LBD HELIX 12 1250 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Kim K et al.,2003 E542Q LBD HELIX 12 1250 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Norris JD et al.,1998 M543A LBD HELIX 12 1251 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Webb P et al.,1999 M543A LBD HELIX 12 1251 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Pearce ST et al.,2003 M543A LBD HELIX 12 1251 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Leone DP et al.,2003 M543A LBD HELIX 12 1251 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Dunn CA et al.,2003 L544A LBD HELIX 12 1252 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Webb P et al.,1999 L544A LBD HELIX 12 1252 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Pearce ST et al.,2003 L544A LBD HELIX 12 1252 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Leone DP et al.,2003 L544A LBD HELIX 12 1252 ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Dunn CA et al.,2003 D545A C-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Liu H et al.,2001 D545A C-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Sathya G et al.,2002 D545A C-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Pearce ST et al.,2003 D545A C-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Gehm BD et al.,2004 D545N C-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Tcherepanova I et al.,2000 D545N C-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Saville B et al.,2002 D545N C-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Kim K et al.,2003 D545N C-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Norris JD et al.,1998 D545V C-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2003 G556L C-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Schwartz JA et al.,2002 G557L C-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Schwartz JA et al.,2002 S559A C-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Schwartz JA et al.,2002 E562A C-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Schwartz JA et al.,2002 Q565P C-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Schwartz JA et al.,2002 A569T C-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Chen Z et al.,2004 Q580L C-term ESR1_HUMAN (P03372) ESR1,ESR, NR3A1 Eng FC et al.,1997 S10A N-term ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Razandi M et al.,2003 R28C N-term ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Stoica GE et al.,2003 S122A N-term ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Lahooti H et al.,1995 E207A DNA_BIND D019 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Jakacka M et al.,2001 E207A DNA_BIND D019 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Kim K et al.,2003 E207G DNA_BIND D019 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Jakacka M et al.,2001 E207G DNA_BIND D019 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Duan WR et al.,2002 E207G DNA_BIND D019 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Kim K et al.,2003 G208A DNA_BIND D020 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Jakacka M et al.,2001 G208A DNA_BIND D020 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Kim K et al.,2003 G208S DNA_BIND D020 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Jakacka M et al.,2001 G208S DNA_BIND D020 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Duan WR et al.,2002 G208S DNA_BIND D020 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Kim K et al.,2003 K210A DNA_BIND D022 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Jakacka M et al.,2001 A227T DNA_BIND D039 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Jakacka M et al.,2001 C241A DNA_BIND D053 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Santagati S et al.,1997 C244A DNA_BIND D056 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Santagati S et al.,1997 S298A HINGE ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Lahooti H et al.,1995 L358A LBD HELIX 3 343 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Mak HY et al.,1999 I362A LBD HELIX 3 347 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Mak HY et al.,1999 I362D LBD HELIX 3 347 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Mak HY et al.,1999 I362R LBD HELIX 3 347 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Jakacka M et al.,2001 K366A LBD HELIX 3 351 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Mak HY et al.,1999 K366A LBD HELIX 3 351 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Schaufele et al.,1999 K366A LBD HELIX 3 351 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Valentine JE et al.,2000 K366D LBD HELIX 3 351 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Mak HY et al.,1999 K366D LBD HELIX 3 351 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Jakacka M et al.,2001 K366L LBD HELIX 3 351 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Mak HY et al.,1999 K366R LBD HELIX 3 351 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Mak HY et al.,1999 F371A Loop 3-4 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Mak HY et al.,1999 F371A Loop 3-4 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Valentine JE et al.,2000 L376A LBD HELIX 4 448 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Mak HY et al.,1999 L376D LBD HELIX 4 448 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Mak HY et al.,1999 V380A LBD HELIX 4 452 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Mak HY et al.,1999 V380A LBD HELIX 4 452 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Mak HY et al.,2001 V380D LBD HELIX 4 452 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Mak HY et al.,1999 V380D LBD HELIX 4 452 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Mak HY et al.,2001 V380H LBD HELIX 4 452 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Mak HY et al.,2001 L383A LBD HELIX 4 455 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Mak HY et al.,1999 L508A LBD HELIX 10-11 1040 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Valentine JE et al.,2000 L508E LBD HELIX 10-11 1040 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Valentine JE et al.,2000 A509E LBD HELIX 10-11 1041 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Valentine JE et al.,2000 L512A LBD HELIX 10-11 1044 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Valentine JE et al.,2000 L512E LBD HELIX 10-11 1044 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Valentine JE et al.,2000 L515A LBD HELIX 10-11 1047 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Valentine JE et al.,2000 L515E LBD HELIX 10-11 1047 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Valentine JE et al.,2000 S516A LBD HELIX 10-11 1048 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Valentine JE et al.,2000 R519A LBD HELIX 10-11 1051 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Valentine JE et al.,2000 H520A LBD HELIX 10-11 1052 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Valentine JE et al.,2000 S522A LBD HELIX 10-11 1054 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Razandi M et al.,2003 N523A LBD HELIX 10-11 1055 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Valentine JE et al.,2000 G525R LBD HELIX 10-11 1057 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Valentine JE et al.,2000 G525R LBD HELIX 10-11 1057 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Coghill E et al.,2001 G525R LBD HELIX 10-11 1057 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Sohal DS et al.,2001 G525R LBD HELIX 10-11 1057 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Weng Z et al.,2002 G525R LBD HELIX 10-11 1057 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Matsui T et al.,2002 G525R LBD HELIX 10-11 1057 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Schwenk F et al.,1998 Y541A LBD HELIX 12 1245 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Valentine JE et al.,2000 Y541A LBD HELIX 12 1245 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 White R et al.,1997 Y541D LBD HELIX 12 1245 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 White R et al.,1997 Y541E LBD HELIX 12 1245 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 White R et al.,1997 Y541F LBD HELIX 12 1245 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 White R et al.,1997 D542A LBD HELIX 12 1246 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Hong H et al.,1997 D542N LBD HELIX 12 1246 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Valentine JE et al.,2000 D542N LBD HELIX 12 1246 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Hong H et al.,1997 D542N LBD HELIX 12 1246 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Schwartz JA et al.,1997 L543A LBD HELIX 12 1247 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Mak HY et al.,1999 L543A LBD HELIX 12 1247 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Valentine JE et al.,2000 L543A LBD HELIX 12 1247 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Jakacka M et al.,2001 L543A LBD HELIX 12 1247 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Mak HY et al.,2001 L543A LBD HELIX 12 1247 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Pearce ST et al.,2003 L543A LBD HELIX 12 1247 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Hong H et al.,1997 L543A LBD HELIX 12 1247 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Thenot S et al.,1997 L543A LBD HELIX 12 1247 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Chuang FM et al.,1997 L543D LBD HELIX 12 1247 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Schwartz JA et al.,1997 L544A LBD HELIX 12 1248 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Mak HY et al.,1999 L544A LBD HELIX 12 1248 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Valentine JE et al.,2000 L544A LBD HELIX 12 1248 ESR1_MOUSE (P19785) Esr1,Esr, Estr, Estra, Nr3a1 Jakacka M et al.,2001 L544A LBD HELIX 12 &nbs